PF-06305591
目录号: A18748
NaV1.8 blocker
PF-06305591 是一种高效且高度选择性的电压门控钠通道 NaV1.8 阻断剂,其 IC50 为 15 nM。具有出色的临床前体外 ADME 和安全性特性。
Discription | PF-06305591 is a potent and highly selective voltage gated sodium channel NaV1.8 blocker, with an IC50 of 15 nM. An excellent preclinical in vitro ADME and safety profile. | ||
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目录号 | A18748 |
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分子式 | C15H22N4O |
分子量 | 274.36 |
CAS号 | 1449473-97-5 |
SMILES | CC(C)(C)C1=CC=C(NC([C@H]([C@@H](C)C(N)=O)N)=N2)C2=C1 |
其他名称 | PF06305591, PF 06305591 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2