PF-4618433
目录号: A13461
PYK2/FAK 抑制剂
PF-4618433 表现出改善的 PYK2 活性,降低的 p38 活性,并且相对于原型药物 BIRB796,具有更优的整体选择性。
Discription | PF-4618433 shows improved PYK2 potency, reduced p38 activity, and superior overall selectivity relative to the prototype BIRB796. | |||||
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Cell Research |
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目录号 | A13461 |
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分子式 | C24H27N7O2 |
分子量 | 445.52 |
CAS号 | 1166393-85-6 |
SMILES | Cc1ccc(cc1)n2c(cc(n2)C(C)(C)C)NC(=O)Nc3cc(n[nH]3)COc4cccnc4 |
其他名称 | PF 4618433, PF4618433 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2