PHA-767491 是一种强效的、ATP竞争性的双重cdc7/cdk9抑制剂(IC50值分别为10和34 nM),可阻止DNA复制的启动。
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生物活性
Discription | PHA-767491 is a potent, ATP-competitive dual cdc7/cdk9 inhibitor (IC50 values are 10 and 34 nM respectively) that prevents initiation of DNA replication. |
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Targets |
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Cell Research |
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产品信息
目录号 | A11164 |
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分子式 | C12H11N3O |
分子量 | 213.24 |
CAS号 | 845714-00-3 |
SMILES | C1CNC(=O)C2=C1NC(=C2)C3=CC=NC=C3 |
其他名称 | PHA767491 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Useful Calculator
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2
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| 购买 845714-00-3 | 845714-00-3 供应商 | 845714-00-3 花费 | 845714-00-3 生产商 | 订购 845714-00-3 | 845714-00-3 代理商