PIK-294
目录号: A10728
PI3K 抑制剂
PIK-294 是一种 PI3 激酶抑制剂,其效力比其母化合物 PIK-293 高出 20 到 60 倍。它是迄今为止报道的最强效的 p110δ-选择性抑制剂 之一。
Discription | PIK-294 is a PI3 Kinase inhibitor that is 20- to 60-fold more potent than the parent compound, PIK-293. It is one of the most potent p110δ-selective inhibitors that has been reported. | ||
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目录号 | A10728 |
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分子式 | C28H23N7O2 |
分子量 | 489.5 |
CAS号 | 900185-02-6 |
SMILES | CC1=C2C(=CC=C1)N=C(N(C2=O)C3=CC=CC=C3C)CN4C5=C(C(=N4)C6=CC(=CC=C6)O)C(=NC=N5)N |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 91 mg/mL (185.89 mM) | |
Water | Insoluble | ||
Ethanol | Insoluble | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 20.43 mL | 102.15 mL | 204.29 mL |
0.5 mM | 4.09 mL | 20.43 mL | 40.86 mL |
1 mM | 2.04 mL | 10.21 mL | 20.43 mL |
5 mM | 0.41 mL | 2.04 mL | 4.09 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2