PIM447 (LGH447)

目录号: A16807

Pim 抑制剂

PIM447 (LGH447)

PIM447 (LGH447) Chemical Structure

CAS NO. 1210608-43-7

PIM447 (LGH447)是一种新型的pan-PIM激酶抑制剂,其PIM1,PIM2,PIM3的Ki值分别为6 pM,18 pM,9 pM。它也抑制GSK3β,PKN1和PKCτ,但效力显着降低,IC50在1-5μM之间(相对于PIM上Ki的差异> 105倍)。

库存: 现货

规格 价格 数量
2 mg
¥ 1,120.00
5 mg
¥ 2,660.00
10 mg
¥ 3,500.00
Warning 产品仅用于科学研究,不针对患者销售,望谅解.
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