主页 /
Cell Metabolism /
PDE /
Pimobendan (Vetmedin)

Pimobendan (Vetmedin)

Name: Pimobendan (Vetmedin)
SKU: A10733

目录号: A10733

PDE 抑制剂

Pimobendan (Vetmedin) Chemical Structure

CAS NO. 74150-27-9

Pimobendan (Vetmedin)是一种钙增敏剂，具有正性肌力和血管舒张作用。它也是磷酸二酯酶III（PDE3）的选择性抑制剂。

库存：现货

规格	价格	数量
5 mg	￥ 840.00
10 mg	￥ 1,400.00
50 mg	￥ 4,060.00
100 mg	￥ 6,860.00
10mM * 1mL in DMSO	￥ 973.00

大包装询价

或

添加到收藏

产品仅用于科学研究，不针对患者销售，望谅解.

产品详情

生物活性

Pimobendan (Vetmedin)是一种钙增敏剂，具有正性肌力和血管舒张作用。它也是磷酸二酯酶III（PDE3）的选择性抑制剂。

靶点信息

PDE3
0.32 μM

溶解度 *

In vitro (25°C)	DMSO	62 mg/mL (185.42 mM)
	Water	Insoluble
	Ethanol	5 mg/mL (14.95 mM)
In vivo	0.5% methylcellulose	28 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	29.9 mL	149.52 mL	299.04 mL
0.5 mM	5.98 mL	29.9 mL	59.81 mL
1 mM	2.99 mL	14.95 mL	29.9 mL
5 mM	0.6 mL	2.99 mL	5.98 mL

*The above data is based on the productmolecular weight 334.4 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A10733
作用机制	Inhibitor (抑制剂)
M. Wt	334.4
Formula	C19H18N4O2
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	74150-27-9
Synonyms	Vetmedin, Acardi, pimobendane
SMILES	CC1CC(=O)NN=C1C2=CC3=C(C=C2)N=C(N3)C4=CC=C(C=C4)OC