PKI-587 ( Gedatolisib )

Name: PKI-587 ( Gedatolisib )
SKU: A11079
Price: 245 CNY
Rating: 5 (1 reviews)

目录号: A11079

PI3K/mTOR 抑制剂

1 篇发表文献

PKI-587 是一种高效的 PI3K/mTOR 激酶抑制剂，能够抑制 PI3K-α, β, γ, δ 各种亚型和 mTOR，其半抑制浓度（IC50）分别为 0.4, 6.0, 5.4, 6.0 和 1.6 nM。

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Grouped product items
规格	价格	库存
1mg	¥245.00	现货
2mg	¥280.00	现货
5mg	¥315.00	现货
10mg	¥595.00	现货
25mg	¥1,330.00	现货
50mg	¥2,485.00	现货
100mg	¥4,585.00	现货
500mg	¥9,695.00	现货
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重要通知：仅供研究使用。我们不向患者销售。

Data Sheet

SDS

顾客使用 Adooq 产品发表的高质量科研文献

Adooq用户使用PKI-587 ( Gedatolisib )发表的1篇文献

Yusuke Murase, .et al. , Oncol Rep, 2022, Apr;47(4):61 PMID: 35088890

生物活性

Discription

PKI-587 is a highly potent PI3K/mTOR kinase inhibitor that inhibits PI3K-α,β,γ, δ isoforms and mTOR with IC50 of 0.4, 6.0, 5.4, 6.0 and 1.6 nM respectively.

Targets

Target	Value

Cell Research

Cell Line	Type	Value	Description	References

产品信息

目录号	A11079
分子式	C32H41N9O4
分子量	615.7
CAS号	1197160-78-3
SMILES	CN(C)C1CCN(CC1)C(=O)C2=CC=C(C=C2)NC(=O)NC3=CC=C(C=C3)C4=NC(=NC(=N4)N5CCOCC5)N6CCOCC6
其他名称	PKI587, Gedatolisib
储存条件	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

溶解性数据

In vitro	DMSO	2 mg/mL (3.24 mM)
	Water	Insoluble
	Ethanol	Insoluble
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	16.24 mL	81.21 mL	162.42 mL
0.5 mM	3.25 mL	16.24 mL	32.48 mL
1 mM	1.62 mL	8.12 mL	16.24 mL
5 mM	0.32 mL	1.62 mL	3.25 mL

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* Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C₁V₁ = C₂V₂

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