PROTACs
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PROTAC ERRα ligand 2
Catalog No. A18939 ERRα inverse agonistPROTAC ERRα ligand 2 is an estrogen-related receptor α (ERRα) inverse agonist with an IC50 of 5.67 nM. PROTAC ERRα ligand 2 (IC50=5.67 nM) displays a ~11-fold improved potency than XCT790 (IC50=61.3 nM). 了解更多 -
cIAP1 Ligand-Linker Conjugates 3
Catalog No. A18985 PROTAC linkercIAP1 Ligand-Linker Conjugates 3 incorporates an IAP ligand for the E3 ubiquitin ligase, and a PROTAC linker. cIAP1 Ligand-Linker Conjugates 3 can be used to design SNIPERs. 了解更多 -
Pomalidomide-PEG4-C-COOH
Catalog No. A13213 PROTAC linkerPomalidomide-PEG4-C-COOH is a synthesized E3 ligase ligand-linker conjugate that incorporates the Pomalidomide based cereblon ligand and 4-unit PEG linker used in PROTAC technology. 了解更多 -
cIAP1 Ligand-Linker Conjugates 5
Catalog No. A18991 PROTAC linkercIAP1 Ligand-Linker Conjugates 5 incorporates an IAP ligand for the E3 ubiquitin ligase, and a PROTAC linker. cIAP1 Ligand-Linker Conjugates 5 can be used to design SNIPERs. 了解更多 -
NH2-C2-NH-Boc
Catalog No. A12192 PROTAC linkerNH2-C2-NH-Boc (PROTAC Linker 22) is a PROTAC linker, which refers to the alkyl chain composition.NH2-C2-NH-Boc can be used in the synthesis of a series of PROTACs. 了解更多 -
Cl-C6-PEG4-O-CH2COOH
Catalog No. A12719 PROTAC linkerCl-C6-PEG4-O-CH2COOH (PROTAC Linker 4) is a PROTAC linker can be used in the synthesis of chloroalkane-containing PROTACs (HaloPROTACs). 了解更多 -
cIAP1 Ligand-Linker Conjugates 12
Catalog No. A18998 PROTAC linkercIAP1 Ligand-Linker Conjugates 12 incorporates an IAP ligand for the E3 ubiquitin ligase, and a PROTAC linker. cIAP1 Ligand-Linker Conjugates 12 can be used to design SNIPERs. 了解更多 -
cIAP1 Ligand-Linker Conjugates 2
Catalog No. A19004 PROTAC linkercIAP1 Ligand-Linker Conjugates 2 incorporates an IAP ligand for the E3 ubiquitin ligase, and a PROTAC linker. cIAP1 Ligand-Linker Conjugates 2 can be used to design SNIPERs. 了解更多 -
cIAP1 Ligand-Linker Conjugates 14
Catalog No. A19010 PROTAC linkercIAP1 Ligand-Linker Conjugates 14 incorporates an IAP ligand for the E3 ubiquitin ligase, and a PROTAC linker. cIAP1 Ligand-Linker Conjugates 14 can be used to design SNIPERs. 了解更多 -
cIAP1 Ligand-Linker Conjugates 15
Catalog No. A19016 PROTAC linkercIAP1 Ligand-Linker Conjugates 15 incorporates an IAP ligand for the E3 ubiquitin ligase, and a PROTAC linker. cIAP1 Ligand-Linker Conjugates 15 can be used to design SNIPERs. 了解更多 -
cIAP1 Ligand-Linker Conjugates 11
Catalog No. A19022 PROTAC linkercIAP1 Ligand-Linker Conjugates 11 incorporates an IAP ligand for the E3 ubiquitin ligase, and a PROTAC linker. cIAP1 Ligand-Linker Conjugates 11 can be used to design SNIPERs. 了解更多 -
Bis-PEG4-acid
Catalog No. A19036 -
Tos-PEG3-O-C1-CH3COO
Catalog No. A19077 PROTAC linkerTos-PEG3-O-C1-CH3COO (PROTAC Linker 6) is a PROTAC linker, which refers to the PEGs composition. 了解更多 -
NH2-PEG3-C1-Boc
Catalog No. A19084 PROTAC linkerNH2-PEG3-C1-Boc (PROTAC Linker 5) is a PROTAC linker, which refers to the PEG composition. NH2-PEG3-C1-Boc can be used in the synthesis of a series of PROTACs. 了解更多 -
cIAP1 Ligand-Linker Conjugates 1
Catalog No. A18978 PROTAC linkercIAP1 Ligand-Linker Conjugates 1 incorporates an IAP ligand for the E3 ubiquitin ligase, and a PROTAC linker. cIAP1 Ligand-Linker Conjugates 1 can be used to design SNIPERs. 了解更多 -
Bis-NH2-PEG2
Catalog No. A18944 PROTAC linkerBis-NH2-PEG2 (PROTAC Linker 19) is a PROTAC linker, which refers to the PEG composition. Bis-NH2-PEG2 can be used in the synthesis of a series of PROTACs. 了解更多 -
VH032-PEG5-C6-Cl
Catalog No. A12884 small molecule HaloPROTACVH032-PEG5-C6-Cl (HaloPROTAC 2) is a small molecule HaloPROTAC that incorporates the VH032 based VHL ligand and 5-unit PEG linker. 了解更多 -
Dox-Ph-PEG1-Cl
Catalog No. A18413 PROTAC linkerDox-Ph-PEG1-Cl (PROTAC Linker 34) is a PROTAC linker, which refers to the PEG composition. Dox-Ph-PEG1-Cl can be used in the synthesis of a series of PROTACs. 了解更多 -
Boc-NH-PEG2-C2-amido-C4-acid
Catalog No. A18425 PROTAC linkerBoc-NH-PEG2-C2-amido-C4-acid (PROTAC Linker 30) is a PROTAC linker, which refers to the PEG composition. Boc-NH-PEG2-C2-amido-C4-acid can be used in the synthesis of a series of PROTACs. 了解更多 -
PEG6-(CH2CO2H)2
Catalog No. A18422 PEG PROTAC linkerPEG6-(CH2CO2H)2 is a PEG derivative containing two terminal carboxylic acid groups. The hydrophilic PEG spacer increases solubility in aqueous media. 了解更多 -
Boc-NH-C6-amido-C4-acid
Catalog No. A18421 PROTAC linkerBoc-NH-C6-amido-C4-acid is a PROTAC linker, which refers to the alkyl/ether composition. Boc-NH-C6-amido-C4-acid can be used in the synthesis of a series of PROTACs. 了解更多 -
NH2-Ph-C4-acid-NH2-Me
Catalog No. A18436 PROTAC linkerNH2-Ph-C4-acid-NH2-Me (PROTAC Linker 31) is a PROTAC linker, which refers to the Alkyl-Chain composition. NH2-Ph-C4-acid-NH2-Me can be used in the synthesis of a series of PROTACs. 了解更多 -
N3-PEG4-C2-NH2
Catalog No. A18938 PROTAC linkerN3-PEG4-C2-NH2 (PROTAC Linker 20) is a polyethylene glycol (PEG)-based PROTAC linker. N3-PEG4-C2-NH2 can be used in the synthesis of a series of PROTACs. 了解更多 -
Phenol-amido-C1-PEG3-N3
Catalog No. A18931 PROTAC linkerPhenol-amido-C1-PEG3-N3 (PROTAC Linker 21) is a PROTAC linker, which refers to the PEG composition. Phenol-amido-C1-PEG3-N3 can be used in the synthesis of a series of PROTACs. 了解更多 -
Tos-PEG4-NH-Boc
Catalog No. A19070 PROTAC linkerTos-PEG4-NH-Boc (PROTAC Linker 7) is a PROTAC linker, which refers to the PEG composition. Tos-PEG4-NH-Boc can be used in the synthesis of a series of PROTACs. 了解更多 -
PEG3-O-CH2COOH
Catalog No. A19063 PROTAC linkerPEG3-O-CH2COOH (Compound 15b) is a PROTAC linker can be used in the synthesis of a series of SNIPER(ER)s. 了解更多 -
Bis-PEG1-C-PEG1-CH2COOH
Catalog No. A18848 PROTAC linkerBis-PEG1-C-PEG1-CH2COOH (PROTAC Linker 26) is a PROTAC linker, which refers to the PEG composition. Bis-PEG1-C-PEG1-CH2COOH can be used in the synthesis of a series of PROTACs. 了解更多 -
Tos-PEG3-NH-Boc
Catalog No. A19057 PROTAC linkerTos-PEG3-NH-Boc (PROTAC Linker 9) is a PROTAC linker, which refers to the PEG composition. Tos-PEG3-NH-Boc can be used in the synthesis of a series of PROTACs. 了解更多 -
Bis-NH2-C1-PEG3
Catalog No. A18870 PROTAC linkerBis-NH2-C1-PEG3 (PROTAC Linker 24) is a PROTAC linker, which refers to the alkyl/ether composition. Bis-NH2-C1-PEG3 can be used in the synthesis of a series of PROTACs. 了解更多