Proxyphylline
目录号: A16821
A1 adenosine receptors 拮抗剂
Proxyphylline 是茶碱的衍生物，用作支气管扩张剂并具有心血管特性。它选择性地拮抗 A1 腺苷受体（Ki = 82 nM，用于牛脑）相比于 A2 腺苷受体（Ki = 850 μM，用于血小板）。
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生物活性
| Discription | Proxyphylline is a derivative of theophylline which is used as a bronchodilator and for its cardiovascular properties. It selectively antagonizes A1 adenosine receptors (Ki = 82 nM for bovine brain) versus A2 adenosine receptors (Ki = 850 μM for platelets). |
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产品信息
| 目录号 | A16821 |
|---|---|
| 分子式 | C10H14N4O3 |
| 分子量 | 238.25 |
| CAS号 | 603-00-9 |
| SMILES | CC(CN1C=NC2=C1C(=O)N(C(=O)N2C)C)O |
| 储存条件 | Store lyophilized at -20ºC, keep desiccated. |
溶解性数据
| In vitro | DMSO | 42 mg/mL (176.29 mM) | |
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* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
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Preparing Stock Solutions
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 41.97 mL | 209.86 mL | 419.73 mL |
| 0.5 mM | 8.39 mL | 41.97 mL | 83.95 mL |
| 1 mM | 4.2 mL | 20.99 mL | 41.97 mL |
| 5 mM | 0.84 mL | 4.2 mL | 8.39 mL |
Useful Calculator
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2
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| 购买 603-00-9 | 603-00-9 供应商 | 603-00-9 花费 | 603-00-9 生产商 | 订购 603-00-9 | 603-00-9 代理商