(Rac)-VU 6008667

Name: (Rac)-VU 6008667
SKU: A21939

目录号: A21939

mAChR M5 negative allosteric modulator

(Rac)-VU 6008667 Chemical Structure

CAS NO. 2092917-63-8

(Rac)-VU 6008667 is a selective negative allosteric modulator of muscarinic acetylcholine receptor subtype 5 (M5 NAM) (IC50=1.8 μM, pIC50= 5.75), has high CNS penetration.

库存：现货

规格	价格	数量
5 mg	￥ 1,134.00
10 mg	￥ 1,953.00
50 mg	￥ 5,796.00
100 mg	￥ 11,592.00

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产品仅用于科学研究，不针对患者销售，望谅解.

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生物活性

(Rac)-VU 6008667 is a selective negative allosteric modulator of muscarinic acetylcholine receptor subtype 5 (M5 NAM) (IC50=1.8 μM, pIC50= 5.75), has high CNS penetration.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	22.79 mL	113.93 mL	227.87 mL
0.5 mM	4.56 mL	22.79 mL	45.57 mL
1 mM	2.28 mL	11.39 mL	22.79 mL
5 mM	0.46 mL	2.28 mL	4.56 mL

*The above data is based on the productmolecular weight 438.85. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A21939
作用机制	Modulator (调节剂)
M. Wt	438.85
Formula	C24H17ClF2N2O2
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	2092917-63-8
Synonyms	VU6008667, VU-6008667
SMILES	O=C1N2C(N(C(C3=CC=C(F)C(F)=C3)=O)CC2)(C4=CC=C(Cl)C(C)=C4)C5=C1C=CC=C5