Ralinepag
目录号: A21073
IP receptor agonist
Ralinepag 是一种强效的、口服生物利用度高的非前列腺素类前列腺素(IP)受体激动剂,其对人类和大鼠 IP 受体以及人类 DP1 受体的 EC50 分别为 8.5 nM、530 nM 和 850 nM。
Discription | Ralinepag is a potent, orally bioavailable and non-prostanoid prostacyclin (IP) receptor agonist, with EC50s of 8.5 nM, 530 nM and 850 nM for human and rat IP receptor and human DP1 receptor, respectively. | ||
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目录号 | A21073 |
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分子式 | C23H26ClNO5 |
分子量 | 431.91 |
CAS号 | 1187856-49-0 |
SMILES | O=C(O)COC[C@H]1CC[C@H](COC(N(C2=CC=C(Cl)C=C2)C3=CC=CC=C3)=O)CC1 |
其他名称 | APD811, APD 811, APD-811 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2