Ruboxistaurin (LY333531 HCl)

Name: Ruboxistaurin (LY333531 HCl)
SKU: A16604

目录号: A16604

PKCβ1 and PKCβ2 抑制剂

Ruboxistaurin (LY333531 HCl) Chemical Structure

CAS NO. 169939-93-9

LY333531是一种特异性β-蛋白激酶C的抑制剂。竞争性和可逆性抑制PKCβ1和PKCβ2，IC50值分别为4.7和5.9 nM。

库存：现货

规格	价格	数量
2 mg	￥ 420.00
5 mg	￥ 700.00
10 mg	￥ 1,540.00
50 mg	￥ 4,060.00

大包装询价

或

添加到收藏

产品仅用于科学研究，不针对患者销售，望谅解.

产品详情

生物活性

LY333531是一种特异性β-蛋白激酶C的抑制剂。竞争性和可逆性抑制PKCβ1和PKCβ2，IC50值分别为4.7和5.9 nM。

溶解度 *

In vitro	DMSO	49 mg/mL (97.02 mM)
	Water	Insoluble
	Ethanol	Insoluble
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	19.8 mL	99.01 mL	198.02 mL
0.5 mM	3.96 mL	19.8 mL	39.6 mL
1 mM	1.98 mL	9.9 mL	19.8 mL
5 mM	0.4 mL	1.98 mL	3.96 mL

*The above data is based on the productmolecular weight 505.01. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A16604
作用机制	Inhibitor (抑制剂)
M. Wt	505.01
Formula	C28H28N4O3.HCl
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	169939-93-9
Synonyms	LY-333531, LY 333531
SMILES	O=C1NC(C2=C1C3=CN(C4=CC=CC=C34)CC[C@@H](CN(C)C)OCCN5C=C2C6=CC=CC=C56)=O.[H]Cl