S1RA (E-52862)
目录号: A12504
sigma-1 receptor 拮抗剂
S1RA 是一种选择性 sigma-1 受体拮抗剂,其报告的结合亲和力为 Ki = 17.0 ± 7.0 nM,相对于 sigma-2 受体 以及其他170种受体、酶、转运蛋白和离子通道具有选择性。
Discription | S1RA is a selective sigma-1 receptor antagonist, with a reported binding affinity of Ki = 17.0 ?? 7.0 nM, selective over the sigma-2 receptor and against a panel of other 170 receptors, enzymes, transporters and ion channels. | |||||
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Targets |
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Cell Research |
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目录号 | A12504 |
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分子式 | C20H23N3O2 |
分子量 | 337.42 |
CAS号 | 878141-96-9 |
SMILES | CC1=CC(=NN1C2=CC3=CC=CC=C3C=C2)OCCN4CCOCC4 |
其他名称 | E52862, E 52862, MR390; MR 390; MR-390 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 63 mg/mL (186.71 mM) | |
Water | 63 mg/mL (186.71 mM) | ||
Ethanol | 18 mg/mL (53.34 mM) | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 29.64 mL | 148.18 mL | 296.37 mL |
0.5 mM | 5.93 mL | 29.64 mL | 59.27 mL |
1 mM | 2.96 mL | 14.82 mL | 29.64 mL |
5 mM | 0.59 mL | 2.96 mL | 5.93 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2