SB-408124 HCl
目录号: A15231
OX Receptor Ant激动剂
SB408124 Hcl 是一种非肽类拮抗剂,针对 OX1 受体,其在整个细胞和膜中的 Ki 分别为 57 nM 和 27 nM;对 OX2 受体显示出 50 倍的选择性。
Discription | SB408124 Hcl is a non-peptide antagonist for OX1 receptor with Ki of 57 nM and 27 nM in both whole cell and membrane, respectively; exhibits 50-fold selectivity over OX2 receptor. | ||
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目录号 | A15231 |
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分子式 | C19H19ClF2N4O |
分子量 | 392.83 |
CAS号 | 1431697-90-3 |
SMILES | CC1=NC2=C(C=C(C=C2C(=C1)NC(=O)NC3=CC=C(C=C3)N(C)C)F)F.Cl |
其他名称 | SB 408124 Hydrochloride, SB408124 Hydrochloride |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2