扫码关注我们
微信二维码

SB-408124

目录号: A11567
OX Receptor Ant激动剂
SB-408124 是一种选择性的非肽类orexin OX1受体拮抗剂(对人类OX1和OX2受体的Kb值分别为21.7和1405 nM)。在体内通过口服给药后,可阻断orexin-A诱导的修饰行为。
Grouped product items
规格 价格 库存 数量
5mg
¥245.00
现货
10mg
¥385.00
现货
25mg
¥805.00
现货
50mg
¥1,435.00
现货
100mg
¥2,625.00
现货
10mM * 1mL in DMSO
¥350.00
现货
更大包装
更多折扣
全国免运费, 顺丰次日达

重要通知:仅供研究使用。我们不向患者销售。

顾客使用 Adooq 产品发表的高质量科研文献
生物活性
Discription SB-408124 is a selective non-peptide orexin OX1 receptor antagonist (Kb values are 21.7 and 1405 nM for human OX1 and OX2 receptors respectively). Blocks orexin-A induced grooming following oral administration in vivo.
Targets
Target Value
产品信息
目录号 A11567
分子式 C19H18F2N4O
分子量 356.37
CAS号 288150-92-5
SMILES CC1=NC2=C(C=C(C=C2C(=C1)NC(=O)NC3=CC=C(C=C3)N(C)C)F)F
其他名称 SB408124, SB 408124
储存条件

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

溶解性数据
In vitro (25°C) DMSO 35 mg/mL (98.2 mM)
Water Insoluble
Ethanol Insoluble
In vivo 30% propylene glycol, 5% Tween 80, 65% D5W 28 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Preparing Stock Solutions
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 28.06 mL 140.3 mL 280.61 mL
0.5 mM 5.61 mL 28.06 mL 56.12 mL
1 mM 2.81 mL 14.03 mL 28.06 mL
5 mM 0.56 mL 2.81 mL 5.61 mL
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

  • Mass

    Concentration

    Volume

    Molecular Weight

Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

  • C1

    V1

    C2

    V2

  • Calculator Reset
Keywords: 购买 SB-408124 | SB-408124 供应商 | SB-408124 花费 | SB-408124 生产商 | 订购 SB-408124 | SB-408124 代理商 | 购买 288150-92-5 | 288150-92-5 供应商 | 288150-92-5 花费 | 288150-92-5 生产商 | 订购 288150-92-5 | 288150-92-5 代理商
苏ICP备14027875号-1