Seclidemstat
目录号: A19730
LSD1 inhibitor
Seclidemstat(SP-2577)是一种效力强大且可口服生物利用度的LSD1抑制剂,平均IC50为127 nM。
Discription | Seclidemstat (SP-2577) is a potent and orally bioavailable LSD1 inhibitor, with a mean IC50 of 127 nM. |
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目录号 | A19730 |
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分子式 | C20H23ClN4O4S |
分子量 | 450.94 |
CAS号 | 1423715-37-0 |
SMILES | O=C(N/N=C(C1=CC(Cl)=CC=C1O)\C)C2=CC=CC(S(=O)(N3CCN(C)CC3)=O)=C2 |
其他名称 | SP-2577, SP2577, SP 2577 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 86 mg/mL (190.71 mM) | |
Water | <1 mg/mL | ||
Ethanol | <1 mg/mL | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 22.18 mL | 110.88 mL | 221.76 mL |
0.5 mM | 4.44 mL | 22.18 mL | 44.35 mL |
1 mM | 2.22 mL | 11.09 mL | 22.18 mL |
5 mM | 0.44 mL | 2.22 mL | 4.44 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2