SHU 9119
目录号: A22734
MC3/4R Antagonist
SHU 9119 是一种强效的人类黑皮素皮质素3和4受体(MC3/4R)拮抗剂,并且是部分MC5R激动剂;其对人类MC3R、MC4R和MC5R的IC50值分别为0.23、0.06和0.09纳摩尔。
MC3/4R Antagonist
Discription | SHU 9119 is a potent human melanocortin 3 and 4 receptors (MC3/4R) antagonist and a partial MC5R agonist; with IC50 values of 0.23, 0.06, and 0.09 nM for human MC3R, MC4R and MC5R, respectively. | |||||
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Cell Research |
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目录号 | A22734 |
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分子式 | C54H71N15O9 |
分子量 | 1074.24 |
CAS号 | 168482-23-3 |
Sequence | Ac-{Nle}-Asp-His-{d-Nal}-Arg-Trp-Lys (Lactam bridge: Asp2-Lys7) |
Sequence shortening | Ac-{Nle}-DH-{d-Nal}-RWK (Lactam bridge: Asp2-Lys7) |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2