Sograzepide
目录号: A22020
Gastrin/CCK-B antagonist
Sograzepide(Netazepide;YF 476;YM-220)是一种极其强效、高度选择性且口服活性的胃泌素/CCK-B拮抗剂,具有0.1 nM的IC50值,对胃泌素/CCK-A活性具有抑制作用,其IC50为502 nM。
Discription | Sograzepide (Netazepide; YF 476; YM-220) is an extremely potent , highly selective and orally active Gastrin/CCK-B antagonist with an IC50 value of 0.1 nM, has inhibitory effect on Gastrin/CCK-A activity with an IC50 of 502 nM. |
---|
目录号 | A22020 |
---|---|
分子式 | C28H30N6O3 |
分子量 | 498.58 |
CAS号 | 155488-25-8 |
SMILES | O=C(NC1=CC=CC(NC)=C1)N[C@H]2C(N(CC(C(C)(C)C)=O)C3=CC=CC=C3C(C4=NC=CC=C4)=N2)=O |
其他名称 | Netazepide; YF 476, YF-476, YF476; YM-220, YM220, YM 220 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2