SR-2211
目录号: A13568
RORr 激动剂
SR-2211 选择性结合 RORr(Ki = 105 nM),作为体外 RORr 活性的反向激动剂(IC50 = 320 nM)。
Discription | SR-2211 selectively binds RORr(Ki = 105 nM), acting as an inverse agonist of constitutive in vitro RORr activity (IC50 = 320 nM). | |||||
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Cell Research |
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目录号 | A13568 |
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分子式 | C26H24F7N3O |
分子量 | 527.5 |
CAS号 | 1359164-11-6 |
SMILES | C1CN(CCN1CC2=CC=C(C=C2)C3=C(C=C(C=C3)C(C(F)(F)F)(C(F)(F)F)O)F)CC4=CC=NC=C4 |
其他名称 | SR 2211, SR2211 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2