SR10067
目录号: A18671
Rev-Erbα/β 激动剂
SR10067 是一种强效、选择性且能穿透大脑的 Rev-Erbα/β 激动剂,其 IC50 值分别针对 Rev-Erbβ 和 Rev-Erbα 为 160 nM 和 170 nM。SR10067 具有抗焦虑活性。
Discription | SR10067 is a potent, selective and brain penetrant Rev-Erbα/β agonist, with IC50 values are 160 and 170 nM for Rev-Erbβ and Rev-Erbα, respectively. SR10067 has anxiolytic activity. |
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目录号 | A18671 |
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分子式 | C31H31NO3 |
分子量 | 465.58 |
CAS号 | 1380548-02-6 |
SMILES | CC(OC1=CC=C(OCC2CC3=CC=CC=C3CN2C(C4=CC=CC5=C4C=CC=C5)=O)C=C1)(C)C |
其他名称 | SR 10067, SR-10067 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2