SSTR5 antagonist 1
目录号: A20218
SSTR5 拮抗剂
SSTR5 antagonist 1 是一种效力强、选择性高、可口服的生长抑素受体亚型 5(SSTR5)拮抗剂,其半抑制浓度(IC50)分别为 9.6 nM 和 57 nM,针对人类 SSTR5(hSSTR5)和小鼠 SSTR5(mSSTR5)。(化合物 25a)。
Discription | SSTR5 antagonist 1 is a potent, selective, and orally available somatostatin receptor subtype 5 (SSTR5) antagonist with IC50s of 9.6 and 57 nM for hSSTR5 and mSSTR5, respectively. (Compound 25a). |
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目录号 | A20218 |
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分子式 | C28H34FN3O5 |
分子量 | 511.59 |
CAS号 | 1628741-91-2 |
SMILES | OC(C1CCN(C2=NOC3(CN(CC4=CC(OCC)=C(C5=CC=C(F)C=C5)C(OCC)=C4)C3)C2)CC1)=O |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2