产品详情

生物活性

SU6656是Src激酶的选择性抑制剂，包括Src，Yes，Lyn和Fyn（分别为IC50 = 280、20、130、170 nM）。

靶点信息

YES	Lyn	Fyn	Src
20 nM	130 nM	170 nM	280 nM

溶解度 *

In vitro (25°C)	DMSO	Warmed: 73 mg/mL (196.52 mM)
	Water	Insoluble
	Ethanol	Insoluble
In vivo	10% DMSO+dd H2O	15 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	26.92 mL	134.61 mL	269.22 mL
0.5 mM	5.38 mL	26.92 mL	53.84 mL
1 mM	2.69 mL	13.46 mL	26.92 mL
5 mM	0.54 mL	2.69 mL	5.38 mL

*The above data is based on the productmolecular weight 371.45. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A15518
作用机制	Inhibitor (抑制剂)
M. Wt	371.45
Formula	C19H21N3O3S
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	330161-87-0
Synonyms	SU-6656, SU 6656
SMILES	CN(C)S(=O)(=O)C1=CC2=C(C=C1)NC(=O)C2=CC3=CC4=C(N3)CCCC4