T338C Src-IN-2
目录号: A16244
Src 抑制剂
T338C Src-IN-2 是一种强效的突变型 c-Src T338C 激酶抑制剂,其 IC50 为 317 nM;同时也能抑制 T338C/V323A 和 T338C/V323S,其 IC50 分别为 57 nM 和 19 nM。
Discription | T338C Src-IN-2 is a potent mutant c-Src T338C kinase inhibitor with IC50 of 317 nM; also inhibits T338C/V323A and T338C/V323S with IC50 of 57 nM/19 nM. |
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目录号 | A16244 |
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分子式 | C17H18FN5O |
分子量 | 327.36 |
CAS号 | 1351927-00-8 |
SMILES | CC(C)N1C2=C(C(=N1)CC3=CC=CC(=C3)C(=O)CF)C(=NC=N2)N |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2