TAK-063
目录号: A15799
PDE10A 抑制剂?€?
TAK-063 是一种高效、选择性和口服活性的 PDE10A 抑制剂，其 IC50 为 0.30 nM；对其他 PDEs 的选择性超过 15000 倍。
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生物活性
| Discription | TAK-063 is a highly potent, selective and orally active PDE10A inhibitor with IC50 of 0.30 nM; >15000-fold selectivity over other PDEs. |
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产品信息
| 目录号 | A15799 |
|---|---|
| 分子式 | C23H17FN6O2 |
| 分子量 | 428.42 |
| CAS号 | 1238697-26-1 |
| SMILES | COC1=CN(N=C(C1=O)C2=CC=NN2C3=CC=CC=C3)C4=C(C=C(C=C4)N5C=CC=N5)F |
| 其他名称 | TAK 063, TAK063 |
| 储存条件 | Store lyophilized at -20ºC, keep desiccated. |
溶解性数据
| In vitro | DMSO | 73 mg/mL (170.39 mM) | |
| Water | Insoluble | ||
| Ethanol | Insoluble | ||
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* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
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Preparing Stock Solutions
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 23.34 mL | 116.71 mL | 233.42 mL |
| 0.5 mM | 4.67 mL | 23.34 mL | 46.68 mL |
| 1 mM | 2.33 mL | 11.67 mL | 23.34 mL |
| 5 mM | 0.47 mL | 2.33 mL | 4.67 mL |
Useful Calculator
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2
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| 购买 1238697-26-1 | 1238697-26-1 供应商 | 1238697-26-1 花费 | 1238697-26-1 生产商 | 订购 1238697-26-1 | 1238697-26-1 代理商