TAK-243

Name: TAK-243
SKU: A20369
Price: 245 CNY
Rating: 5 (288 reviews)

目录号: A20369

UAE (UBA1) 抑制剂

TAK-243 (MLN7243) 是一种首创的、选择性的泛素激活酶（UAE，UBA1）抑制剂（IC50=1 nM），它阻断泛素连接，打断单泛素信号传递以及全局蛋白质泛素化。

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Grouped product items
规格	价格	库存
1mg	¥245.00	现货
2mg	¥350.00	现货
5mg	¥630.00	现货
10mg	¥1,015.00	现货
25mg	¥1,925.00	现货
50mg	¥3,325.00	现货
100mg	¥4,795.00	现货
*10mM 1mL in DMSO**	¥700.00	现货
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重要通知：仅供研究使用。我们不向患者销售。

Data Sheet

SDS

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生物活性

Discription	TAK-243 (MLN7243) is a first-in-class, selective ubiquitin activating enzyme, UAE (UBA1) inhibitor (IC50=1 nM), which blocks ubiquitin conjugation, disrupting monoubiquitin signaling as well as global protein ubiquitination.

产品信息

目录号	A20369
分子式	C19H20F3N5O5S2
分子量	519.52
CAS号	1450833-55-2
SMILES	O=S(OC[C@@H]1[C@@H](O)[C@@H](O)[C@H](NC2=CC=NC3=CC(C4=CC=CC(SC(F)(F)F)=C4)=NN23)C1)(N)=O
其他名称	TAK 243, TAK243, MLN7243, MLN 7243, MLN-7243
储存条件	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

溶解性数据

In vitro	DMSO	85 mg/mL (163.61 mM)
	Water	Insoluble
	Ethanol	21 mg/mL (40.42 mM)
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	19.25 mL	96.24 mL	192.49 mL
0.5 mM	3.85 mL	19.25 mL	38.5 mL
1 mM	1.92 mL	9.62 mL	19.25 mL
5 mM	0.38 mL	1.92 mL	3.85 mL

Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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* Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C₁V₁ = C₂V₂

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