TAS-115 mesylate
目录号: A21389
c-Met/HGFR 抑制剂
TAS-115 mesylate 是一种强效的 VEGFR 和肝细胞生长因子受体(c-Met/HGFR)靶向激酶抑制剂,其对 rVEGFR2 和 rMET 的 IC50 分别为 30 nM 和 32 nM。
Discription | TAS-115 mesylate is a potent VEGFRand hepatocyte growth factor receptor (c-Met/HGFR)-targeted kinase inhibitor, with IC50s of 30 and 32 nM for rVEGFR2 and rMET, respectively. |
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目录号 | A21389 |
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分子式 | C28H27FN4O7S2 |
分子量 | 614.66 |
CAS号 | 1688673-09-7 |
SMILES | CS(=O)(O)=O.O=C(C1=C(OC)C=C2N=CC=C(OC3=CC=C(NC(NC(CC4=CC=CC=C4)=O)=S)C=C3F)C2=C1)NC |
其他名称 | TAS-115 methanesulfonate, TAS115, TAS 115 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2