TCPOBOP
目录号: A18376
Androstane receptor agonist
TCPOBOP 是一种组成型雄烷酮受体(CAR)的激动剂(EC50 = 20 nM)。TCPOBOP 作为 CAR 的剂量依赖性直接激动剂,增强了核受体CAR对细胞色素P450(CYP)的转录激活。
Discription | TCPOBOP is an agonist of the constitutive androstane receptor (CAR) (EC50 = 20 nM). TCPOBOP enhances the nuclear receptor CAR transactivation of cytochrome P450 (CYP), as dose-dependent direct agonist of CAR. | ||
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目录号 | A18376 |
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分子式 | C16H8Cl4N2O2 |
分子量 | 402.05 |
CAS号 | 76150-91-9 |
SMILES | ClC1=CN=C(OC2=CC=C(OC3=NC=C(Cl)C=C3Cl)C=C2)C(Cl)=C1 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2