Tegaserod maleate
目录号: A11743
5-HT 拮抗剂
Tegaserod 作为一种运动性刺激剂，通过激活胃肠道内脏神经系统中的 5-HT4 受体 来实现其期望的治疗效果。它还刺激胃肠运动和蠕动反射，并据称减少腹痛。此外，tegaserod 是一种 5-HT2B 受体拮抗剂。
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生物活性
| Discription | Tegaserod functions as a motility stimulant, achieving its desired therapeutic effects through activation of the 5-HT4 receptors of the enteric nervous system in the gastrointestinal tract. It also stimulates gastrointestinal motility and the peristaltic reflex, and allegedly reduces abdominal pain. Additionally, tegaserod is a 5-HT2B receptor antagonist. | ||
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产品信息
| 目录号 | A11743 |
|---|---|
| 分子式 | C16H23N5O.C4H4O4 |
| 分子量 | 417.46 |
| CAS号 | 189188-57-6 |
| SMILES | CCCCCN=C(N)NN/C=C/1\C=NC2=C1C=C(C=C2)OC.C(=C\C(=O)O)\C(=O)O |
| 其他名称 | Zelnorm |
| 储存条件 | Store lyophilized at -20ºC, keep desiccated. |
溶解性数据
| In vitro | DMSO | 72 mg/mL (172.47 mM) | |
| Water | Insoluble | ||
| Ethanol | 7 mg/mL (16.77 mM) | ||
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* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
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Preparing Stock Solutions
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 23.95 mL | 119.77 mL | 239.54 mL |
| 0.5 mM | 4.79 mL | 23.95 mL | 47.91 mL |
| 1 mM | 2.4 mL | 11.98 mL | 23.95 mL |
| 5 mM | 0.48 mL | 2.4 mL | 4.79 mL |
Useful Calculator
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2
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| 购买 189188-57-6 | 189188-57-6 供应商 | 189188-57-6 花费 | 189188-57-6 生产商 | 订购 189188-57-6 | 189188-57-6 代理商