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Teneligliptin hydrobromide

Teneligliptin hydrobromide

Name: Teneligliptin hydrobromide
SKU: A15258

目录号: A15258

DPP-4 抑制剂

Teneligliptin hydrobromide Chemical Structure

CAS NO. 906093-29-6

Teneligliptin hydrobromide是一种新颖，有效且持久的二肽基肽酶-4抑制剂。在体外竞争性抑制人血浆，大鼠血浆和人重组DPP-4，IC50值约为1 nM。

库存：现货

规格	价格	数量
100 mg	￥ 1,680.00
200 mg	￥ 3,080.00

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产品仅用于科学研究，不针对患者销售，望谅解.

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生物活性

Teneligliptin hydrobromide是一种新颖，有效且持久的二肽基肽酶-4抑制剂。在体外竞争性抑制人血浆，大鼠血浆和人重组DPP-4，IC50值约为1 nM。

靶点信息

Dipeptidyl peptidase-4	DPP-9	DPP-8	FAP
1.75 nM	150 nM	189 nM	>10 μM

溶解度 *

In vitro	DMSO	85 mg/mL (135.16 mM)
	Water	85 mg/mL (135.16 mM)
	Ethanol	14 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

制备储备液

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	7.95 mL	39.75 mL	79.51 mL
0.5 mM	1.59 mL	7.95 mL	15.9 mL
1 mM	0.8 mL	3.98 mL	7.95 mL
5 mM	0.16 mL	0.8 mL	1.59 mL

*The above data is based on the productmolecular weight 1257.72. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

化学数据

目录号	A15258
作用机制	Inhibitor (抑制剂)
M. Wt	1257.72
Formula	C44H65Br5N12O2S2
Purity	>99%
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.
CAS No.	906093-29-6
SMILES	CC1=NN(C(=C1)N2CCN(CC2)C3CC(NC3)C(=O)N4CCSC4)C5=CC=CC=C5.CC1=NN(C(=C1)N2CCN(CC2)C3CC(NC3)C(=O)N4CCSC4)C5=CC=CC=C5.Br.Br.Br.Br.Br