Teneligliptin
目录号: A15505
DPP-4 抑制剂
Teneligliptin 是一种新型、高效、持久的二肽基肽酶-4抑制剂;在体外竞争性抑制人类血浆、大鼠血浆和人类重组DPP-4,IC50值约为1纳摩尔。
Discription | Teneligliptin is a novel, potent, and long-lasting dipeptidyl peptidase-4 inhibitor; competitively inhibited human plasma, rat plasma, and human recombinant DPP-4 in vitro, with IC50 values of approximately 1 nM. |
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目录号 | A15505 |
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分子式 | C22H30N6OS |
分子量 | 426.58 |
CAS号 | 760937-92-6 |
SMILES | CC1=NN(C(=C1)N2CCN(CC2)C3CC(NC3)C(=O)N4CCSC4)C5=CC=CC=C5 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2