TGR-1202 (Umbralisib)

Name: TGR-1202 (Umbralisib)
SKU: A16277
Price: 245 CNY
Rating: 5 (288 reviews)

目录号: A16277

PI3Kδ inhibitor

TGR-1202 是一种口服的新一代 PI3Kδ 抑制剂，在酶和细胞基础的测定中抑制 PI3Kδ 活性，其 IC50 和 EC50 值分别为 22.2 和 24.3 nM。

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Grouped product items
规格	价格	库存
1mg	¥245.00	现货
2mg	¥350.00	现货
5mg	¥630.00	现货
10mg	¥1,190.00	现货
25mg	¥2,485.00	现货
50mg	¥3,255.00	现货
100mg	¥4,795.00	现货
*10mM 1mL in DMSO**	¥805.00	现货
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Data Sheet

SDS

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生物活性

Discription

TGR-1202 is an orally available, next generation PI3Kδ inhibitor, inhibits PI3Kδ activity in enzyme and cell based assays with IC50 and EC50 values of 22.2 and 24.3 nM respectively.

Targets

Target	Value

产品信息

目录号	A16277
分子式	C31H24F3N5O3
分子量	571.55
CAS号	1532533-67-7
SMILES	CC(C)OC1=C(C=C(C=C1)C2=NN(C3=C2C(=NC=N3)N)C(C)C4=C(C(=O)C5=C(O4)C=CC(=C5)F)C6=CC(=CC=C6)F)F
其他名称	RP5264, TGR1202, TGR 1202, RP-5264, RP 5264
储存条件	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

溶解性数据

In vitro (25°C)	DMSO	Warmed: 92 mg/mL (160.96 mM)
	Water	Insoluble
	Ethanol	Warmed: 6 mg/mL
In vivo	2% DMSO+30% PEG 300+2% Tween 80+H2O	2 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	17.5 mL	87.48 mL	174.96 mL
0.5 mM	3.5 mL	17.5 mL	34.99 mL
1 mM	1.75 mL	8.75 mL	17.5 mL
5 mM	0.35 mL	1.75 mL	3.5 mL

Useful Calculator

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Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C₁V₁ = C₂V₂

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