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TGR-1202是口服的下一代PI3Kδ抑制剂，在基于酶和细胞的测定中抑制PI3Kδ活性，IC50和EC50值分别为22.2和24.3 nM。
| In vitro (25°C) | DMSO | Warmed: 92 mg/mL (160.96 mM) | |
| Water | Insoluble | ||
| Ethanol | Warmed: 6 mg/mL | ||
| In vivo | 2% DMSO+30% PEG 300+2% Tween 80+H2O | 2 mg/mL | |
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
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| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 17.5 mL | 87.48 mL | 174.96 mL |
| 0.5 mM | 3.5 mL | 17.5 mL | 34.99 mL |
| 1 mM | 1.75 mL | 8.75 mL | 17.5 mL |
| 5 mM | 0.35 mL | 1.75 mL | 3.5 mL |
*The above data is based on the productmolecular weight 571.55. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| 目录号 | A16277 |
|---|---|
| 作用机制 | Inhibitor (抑制剂) |
| M. Wt | 571.55 |
| Formula | C31H24F3N5O3 |
| Purity | >99% |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
| CAS No. | 1532533-67-7 |
| Synonyms | RP5264, TGR1202, TGR 1202, RP-5264, RP 5264 |
| SMILES | CC(C)OC1=C(C=C(C=C1)C2=NN(C3=C2C(=NC=N3)N)C(C)C4=C(C(=O)C5=C(O4)C=CC(=C5)F)C6=CC(=CC=C6)F)F |
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