TPCA-1

Name: TPCA-1
SKU: A11579
Price: 210 CNY
Rating: 5 (1 reviews)

目录号: A11579

IKK-2 抑制剂

1 篇发表文献

TPCA-1 是一种针对人类 IκB 激酶-2 (IKK-2) 的强效和选择性抑制剂，其对 IKK-2 的半抑制浓度（IC50）为 17.9 nM，相比之下，对 IKK-1 的 IC50 为 400 nM。

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Grouped product items
规格	价格	库存
2mg	¥210.00	现货
5mg	¥350.00	现货
10mg	¥595.00	现货
25mg	¥1,155.00	现货
50mg	¥1,855.00	现货
100mg	¥2,905.00	现货
*10mM 1mL in DMSO**	¥560.00	现货
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重要通知：仅供研究使用。我们不向患者销售。

Data Sheet

SDS

顾客使用 Adooq 产品发表的高质量科研文献

Adooq用户使用TPCA-1发表的1篇文献

Dongdong Fang, etc. Epithelial-Mesenchymal Transition of Ovarian Cancer Cells Is Sustained by Rac1 through Simultaneous Activation of MEK1/2 and Src Signaling Pathways. Oncogene. 2017 Mar; 36(11): 1546?€?1558.

生物活性

Discription

TPCA-1 is a potent and selective inhibitor of human IκB kinase-2 (IKK-2) with IC50 = 17.9 nM for IKK-2 compared to 400nm for IKK-1.

Targets

Target	Value

产品信息

目录号	A11579
分子式	C12H10FN3O2S
分子量	279.29
CAS号	507475-17-4
SMILES	C1=CC(=CC=C1C2=CC(=C(S2)NC(=O)N)C(=O)N)F
其他名称	TPCA1
储存条件	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

溶解性数据

In vitro (25°C)	DMSO	49 mg/mL (175.44 mM)
	Water	Insoluble
	Ethanol	Insoluble
In vivo	2% Cremophor EL, 2% N,N-dimethylacetamide	14 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	35.81 mL	179.03 mL	358.05 mL
0.5 mM	7.16 mL	35.81 mL	71.61 mL
1 mM	3.58 mL	17.9 mL	35.81 mL
5 mM	0.72 mL	3.58 mL	7.16 mL

Useful Calculator

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* Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C₁V₁ = C₂V₂

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