UM-164
目录号: A19895
c-Src inhibitor
UM-164(DAS-DFGO-II)是一种高效的c-Src抑制剂,其Kd值为2.7 nM。UM-164还能强效抑制p38α和p38β。
Discription | UM-164 (DAS-DFGO-II) is a highly potent inhibitor of c-Src with a Kd of 2.7 nM. UM-164 also potently inhibits p38α and p38β. | ||
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Targets |
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目录号 | A19895 |
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分子式 | C30H31F3N8O3S |
分子量 | 640.68 |
CAS号 | 903564-48-7 |
SMILES | O=C(C1=CN=C(NC2=NC(C)=NC(N3CCN(CCO)CC3)=C2)S1)NC4=CC(NC(C5=CC=CC(C(F)(F)F)=C5)=O)=CC=C4C |
其他名称 | DAS-DFGO-II, UM164, UM 164 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 85 mg/mL (132.67 mM) | |
Water | Insoluble | ||
Ethanol | Insoluble | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 15.61 mL | 78.04 mL | 156.08 mL |
0.5 mM | 3.12 mL | 15.61 mL | 31.22 mL |
1 mM | 1.56 mL | 7.8 mL | 15.61 mL |
5 mM | 0.31 mL | 1.56 mL | 3.12 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2