UNC0646
目录号: A13194
G9a/GLP HMTase 抑制剂
UNC0646 是一种强效且选择性的同源蛋白赖氨酸甲基转移酶 G9a 和 GLP 的抑制剂(IC50 值分别为 G9a 的 6 nM 和 GLP 的 15 nM)。
Discription | UNC0646 is a potent and selective inhibitor of the homologous protein lysine methyltransferases, G9a and GLP (IC50 values are 6 nM and 15 nM for G9a and GLP, respectively). | |||||
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Targets |
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Cell Research |
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目录号 | A13194 |
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分子式 | C36H59N7O2 |
分子量 | 621.9 |
CAS号 | 1320288-17-2 |
SMILES | CC(C)N1CCCN(CC1)C2=NC3=CC(=C(C=C3C(=N2)NC4CCN(CC4)C5CCCCC5)OC)OCCCN6CCCCC6 |
其他名称 | UNC 0646, UNC-0646 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
In vitro | DMSO | 31 mg/mL (49.84 mM) | |
Water | Insoluble | ||
Ethanol | 47 mg/mL | ||
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
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0.1 mM | 16.08 mL | 80.4 mL | 160.8 mL |
0.5 mM | 3.22 mL | 16.08 mL | 32.16 mL |
1 mM | 1.61 mL | 8.04 mL | 16.08 mL |
5 mM | 0.32 mL | 1.61 mL | 3.22 mL |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2