UNC569
目录号: A13805
Mer 抑制剂
UNC569 是一种新型小分子 MER 抑制剂,对体外和体内的急性淋巴细胞性白血病具有疗效。UNC569 是首个小分子 Mer 抑制剂。UNC569 抑制了 Mer 激活及其通过 ERK1/2 和 AKT 的下游信号传导。
Discription | UNC569 is a novel small-molecule MER inhibitor with efficacy against acute lymphoblastic leukemia in vitro and in vivo. UNC569 is the first small-molecule Mer inhibitor. UNC569 inhibited Mer activation and downstream signaling through ERK1/2 and AKT. | |||||
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Cell Research |
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目录号 | A13805 |
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分子式 | C22H29FN6 |
分子量 | 396.5 |
CAS号 | 1350547-65-7 |
SMILES | CCCCNC1=NC=C2C(=NN(C2=N1)CC3CCC(CC3)N)C4=CC=C(C=C4)F |
其他名称 | UNC-569, UNC 569 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2