VER-246608
目录号: A22015
PDK inhibitor
VER-246608 是一种强效且与ATP竞争的丙酮酸脱氢酶激酶(PDK)抑制剂,其半抑制浓度(IC50)分别为针对 PDK-1、PDK-3、PDK-2 和 PDK-4 的 35 nM、40 nM、84 nM 和 91 nM。
Discription | VER-246608 is a potent and ATP-competitive inhibitor of pyruvate dehydrogenase kinase (PDK) with IC50s of 35 nM, 40 nM, 84 nM, and 91 nM for PDK-1, PDK-3, PDK-2, and PDK-4, respectively. | |||||
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Cell Research |
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目录号 | A22015 |
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分子式 | C28H23ClF2N4O4 |
分子量 | 552.96 |
CAS号 | 1684386-71-7 |
SMILES | O=C(C1=CC=C(O)C=C1O)N(CC2=CC=C(CNC(C(F)F)=O)C=C2)C(C=C3)=CC=C3C4=NC(Cl)=NC=C4C |
其他名称 | VER246608, VER 246608 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2