VTP50469
目录号: A22238
Menin-MLL interaction 抑制剂
VTP50469 是一种效力强大、高度选择性且可口服的 Menin-MLL 交互作用抑制剂,其Ki值为104 pM。VTP50469 具有强大的抗白血病活性。
Discription | VTP50469 is a potent, highly selective and orally active Menin-MLL interaction inhibitor with a Ki of 104 pM. VTP50469 has potently anti-leukemia activity. |
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目录号 | A22238 |
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分子式 | C32H47FN6O4S |
分子量 | 630.82 |
CAS号 | 2169916-18-9 |
SMILES | O=C(N(C(C)C)C(C)C)C1=CC(F)=CC=C1OC2=CN=CN=C2N3CC4(CCN(C[C@H]5CC[C@H](NS(=O)(C)=O)CC5)CC4)C3 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2