VU6005649
目录号: A17023
CNS penetrant mGlu7/8 receptor 激动剂
VU6005649 是一种能穿透中枢神经系统(CNS)的 mGlu7/8 受体激动剂,其对 mGlu7 受体和 mGlu8 受体的半最大有效浓度(EC50)分别为 0.65 微米和 2.6 微米。
Discription | VU6005649 is a CNS penetrant mGlu7/8 receptor agonist with EC50s of 0.65 μM and 2.6 μM for mGlu7 receptor and mGlu8 receptor, respectively. | ||
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目录号 | A17023 |
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分子式 | C16H12F5N3O |
分子量 | 357.27 |
CAS号 | 2137047-43-7 |
SMILES | CC1=NN2C(N=C(C)C=C2C(F)(F)F)=C1C3=CC=C(OC)C(F)=C3F |
其他名称 | VU 6005649, VU-6005649 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2