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XE 991 dihydrochloride

目录号: A20032
Kv7 (KCNQ) channels blocker
XE 991 二盐酸盐是一种 Kv7 (KCNQ) 通道阻断剂,能强效抑制 Kv7.1 (KCNQ1)Kv7.2 (KCNQ2)Kv7.2 + Kv7.3 (KCNQ3) 通道以及 M电流,其半抑制浓度(IC50)分别为0.75 μM、0.71 μM、0.6 μM 和 0.98 μM。
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规格 价格 库存 数量
1mg
¥245.00
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5mg
¥630.00
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10mg
¥1,050.00
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25mg
¥2,030.00
现货
50mg
¥3,780.00
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100mg
¥5,530.00
现货
10mM * 1mL in DMSO
¥630.00
现货
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生物活性
Discription XE 991 dihydrochloride, a Kv7 (KCNQ) channels blocker, potently inhibits Kv7.1 (KCNQ1), Kv7.2 (KCNQ2), Kv7.2 + Kv7.3 (KCNQ3) channel, and M-current with IC50s of 0.75 ?M, 0.71 ?M, 0.6 μM, and 0.98 ?M, respectively.
产品信息
目录号 A20032
分子式 C26H22Cl2N2O
分子量 449.37
CAS号 122955-13-9
SMILES O=C1C2=C(C=CC=C2)C(CC3=CC=NC=C3)(CC4=CC=NC=C4)C5=CC=CC=C15.Cl.Cl
其他名称 XE991, XE991
储存条件

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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