XY101
目录号: A18437
RORγ inverse 激动剂
XY101 是一种效力强大、选择性高、代谢稳定且可口服的 RORγ 逆向激动剂,其 IC50 为 30 nM,Kd 为 380 nM。
Discription | XY101 is a potent, selective, metabolically stable and orally available RORγ inverse agonist with an IC50 of 30 nM and a Kd of 380 nM. | |||||
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Cell Research |
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目录号 | A18437 |
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分子式 | C25H20F7NO4S |
分子量 | 563.48 |
CAS号 | 2349368-16-5 |
SMILES | O=S(C1=CC=C(CC(NC2=CC=C(C3=C(F)C=C(C(O)(C(F)(F)F)C(F)(F)F)C=C3)C=C2)=O)C=C1)(CC)=O |
其他名称 | XY 101, XY-101 |
储存条件 | Store lyophilized at -20ºC, keep desiccated. |
Calculate the dilution required to prepare a stock solution. This equation is commonly abbreviated as: C1V1 = C2V2