BTK

Inhibitory Selectivity

Catalog No.	Inhibitor Name	BTK	Other
A11020	Ibrutinib	****	BLK,Bmx,FGR
A13202	AVL-292	****	YES,c-Src,BRK
A13233	CNX-774	***
A15558	ONO-4059 analogue	**
A16261	LFM-A13	*
A12535	RN486	**
A11348	CGI1746	***
A12706	GDC-0834	**
A15008	AVL-292 benzenesulfonate	****	YES,c-Src,BRK
A15824	ACP-196 (Acalabrutinib)	**
A15976	Olmutinib (HM71224)	***
A16262	PCI 29732	**
A16263	QL47	**

Notes:
1.Hover mouse over " * " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " * " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.

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MT-802

Catalog No. A18589
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BTK degrader

MT-802 is a potent BTK degrader based on PROTAC technology, with a DC50 of 1 nM. MT-802 has potential to treat C481S mutant chronic lymphocytic leukemia (CLL). 了解更多

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