Syk
Catalog No. | Inhibitor Name | Syk | Other |
---|---|---|---|
A10769 | R406 besylate | ** | Flt3 |
A10770 | R406 (Tamatinib) | ** | Flt3 |
A10771 | R788 Disodium | ** | |
A12731 | PRT062607 HCl | **** | FGR,MLK1,YES |
A11926 | Fostamatinib | ** | Adenosine A3 receptor,Adenosine transporter,Monoamine transporter |
A16240 | MNS | * | p97,Src |
A15524 | PRT-060318 | **** | |
A13884 | Entospletinib | *** | |
A11320 | BAY-61-3606 | *** | |
A12162 | Piceatannol | Lyn,PKA,PKC | |
A11952 | P505-15 (PRT062607, BIIB057) | **** | FGR, MLK1 |
A14161 | R112 | * |
Notes:
1.Hover mouse over " " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.
-
R406 besylate
Catalog No. A10769 Syk 抑制剂R406 besylate是一种口服酪氨酸激酶抑制剂,IC50为41 nM。对Syk抑制作用强,但是不抑制Lyn,对Flt3的作用比对Syk低5倍。 了解更多