ROCK

Inhibitory Selectivity

Catalog No.	Inhibitor Name	ROCK	ROCK1	ROCK2	Other
A11001	Y-27632 2HCl		*	*
A10928	Thiazovivin	*
A10381	Fasudil HCl			*	PKA,PKG,PKC
A10441	GSK429286A		***	**
A13067	RKI-1447		***	***
A12348	GSK269962		****	****	MSK1,RSK1
A15888	Ripasudil		**	**
A15239	KD025			**
A12464	AT13148		***	****	PKA,p70S6K,Akt1

Notes:
1.Hover mouse over " * " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " * " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.