FLT3

Inhibitory Selectivity

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Catalog No.	Inhibitor Name	FLT3	Other
A10027	Quizartinib	***
A10198	Dovitinib Dilactic Acid	****	c-Kit,FGFR1,VEGFR3/FLT4
A10352	ENMD-2076	***	RET,Aurora A,VEGFR3/FLT4
A10352	ENMD-2076 L-(*)-Tartaric acid		RET,Aurora A,VEGFR3/FLT4
A10508	KW-2449	****	Abl (T315I),Abl,FGFR1
A10610	Amuvatinib	*	c-Kit (D816H),PDGFRα (V561D)
A10769	R406		Syk
A10887	Tandutinib	*	c-Kit,PDGFRβ,CSF-1R
A10996	Cabozantinib	**	VEGFR2/KDR,c-Met,Kit
A11180	TG101209	*	JAK2,RET,JAK3

Showing 1 to 10 of 24 entries

Notes:
1.Hover mouse over " * " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " * " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.

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UNC-2025

Catalog No. A15904
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Dual MER/FLT3 抑制剂

UNC-2025是一种有效的且可生物利用的双重MER/FLT3抑制剂，IC50分别为0.74 nM和0.8 nM，选择性是Axl和Tyro3的20倍。了解更多

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