PDK1

Inhibitory Selectivity

Catalog No.	Inhibitor Name	PDK-1	Other Targets
A10681	OSU-03012	**
A11148	BX-795	****	TBK1/IKKɛ,c-Kit,CDK2/CyclinE
A11149	BX-912	***	PKA,KDR,CDK2/CyclinE
A11032	PHT-427	*	Akt
A12767	GSK2334470	***
A12881	BX-517	****
A11511	NVP-BAG956	*	PI3K
A13484	PS 48	*

Notes:
1.Hover mouse over " * " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " * " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.

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PS 48

Catalog No. A13484
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PDK1 抑制剂

PS 48是一种变构磷酸肌醇依赖性蛋白激酶-1（PDK1）激活剂（Kd = 10.3μM）。了解更多

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TEPP-46

Catalog No. A16279
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PKM2 activator

TEPP-46是重组丙酮酸激酶M2（PKM2）的有效选择性活化剂，最大活化浓度（AC50值）的一半为92 nM，相对于PKM1，PKL和PKR几乎没有或没有活性。了解更多

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