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￥ 0.00 PDK1
| Catalog No. | Inhibitor Name | PDK-1 | Other Targets |
|---|---|---|---|
| A10681 | OSU-03012 | ** | |
| A11148 | BX-795 | **** | TBK1/IKKɛ,c-Kit,CDK2/CyclinE |
| A11149 | BX-912 | *** | PKA,KDR,CDK2/CyclinE |
| A11032 | PHT-427 | * | Akt |
| A12767 | GSK2334470 | *** | |
| A12881 | BX-517 | **** | |
| A11511 | NVP-BAG956 | * | PI3K |
| A13484 | PS 48 | * |
Notes:
1.Hover mouse over "" to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of "" is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.
10 个项目
每页
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PDK1 inhibitor
Catalog No. A11528 -
PDK1 inhibitor
Catalog No. A16185 PDK1 抑制剂PDK1 inhibitor，强效，ATP竞争性和选择性双重PI3K和PDPK1抑制剂（PDK1和p-T308-PKB抑制的IC50值分别为34 nM和94 nM。 了解更多 -
PHT-427
Catalog No. A11032 -
NVP-BAG956
Catalog No. A11511 PI3K/PDK-1 抑制剂NVP-BAG956是一种强效、可逆和ATP竞争性PI3-K/PDK1双激酶抑制剂，对VEGFR 1(IC50 = 2.56 μM)的效力大大降低，对其他15种激酶(IC50 > 10 uM)的活性很小或没有活性。 了解更多 -
GSK 2334470
Catalog No. A12767 -
BX-517
Catalog No. A12881
10 个项目
每页