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￥ 0.00 COX
| Catalog No. | Inhibitor Name | COX | COX-1 | COX-2 | Other |
|---|---|---|---|---|---|
| A10193 | Celecoxib | **** | |||
| A10461 | Ibuprofen | * | * | ||
| A10474 | Indomethacin | ** | * | ||
| A11918 | Rofecoxib | **** | |||
| A10304 | Diclofenac Sodium | *** | *** | ||
| A11695 | Lornoxicam | **** | **** | ||
| A10623 | Naproxen Sodium | * | * | ||
| A13342 | Valdecoxib | **** | |||
| A11693 | Tolfenamic Acid | *** | |||
| A16399 | Amfenac Sodium Monohydrate | ** | *** | ||
| A11694 | Nimesulide | * | |||
| A12520 | Meclofenamate Sodium | **** | *** | ||
| A16428 | Carprofen | **** | |||
| A10636 | Nepafenac | ||||
| A10878 | Sulindac | ||||
| A10565 | Meloxicam | ||||
| A10820 | Aspirin | ||||
| A11906 | Phenacetin | ||||
| A10736 | Piroxicam | ||||
| A10462 | Ibuprofen Lysine | ||||
| A11641 | Pranoprofen | ||||
| A10090 | Asaraldehyde | ||||
| A11692 | Acemetacin | ||||
| A13244 | Bromfenac Sodium |
Notes:
1.Hover mouse over "" to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of "" is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.
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Bromfenac sodium
Catalog No. A13244 -
Acetaminophen
Catalog No. A10030 COX 抑制剂Acetaminophen (paracetamol) 是选择性环氧合酶-2 (COX-2) 的抑制剂，IC50 值为 25.8 μM。Acetaminophen 是一种有效的肝 N-乙酰转移酶 2 (NAT2) 抑制剂。它是广泛使用的解热和止痛药。 了解更多 -
Naproxen sodium
Catalog No. A10623 COX 抑制剂Naproxen sodium是一种非选择性的环氧合酶（COX）抑制剂，具有抗炎，解热和镇痛作用。对秋水仙碱引起的认知障碍和氧化应激具有神经保护作用。 了解更多 -
FK 3311
Catalog No. A13332 -
Valdecoxib
Catalog No. A13342 COX-2 抑制剂伐地考昔（Valdecoxib），也称为SC-65872，是一种非甾体类抗炎药（NSAID），用于治疗骨关节炎，类风湿性关节炎以及痛经和月经症状。 它是一种选择性的环氧合酶2（COX-2)抑制剂,IC50为5nM。 了解更多 -
Amfenac Sodium Monohydrate
Catalog No. A16399 COX 抑制剂Amfenac Sodium Monohydrate是一种非甾体止痛消炎药，带有乙酸部分。COX1和COX2的IC50值分别为250 nM和150 nM。 了解更多 -
Carprofen
Catalog No. A16428 -
Timegadine
Catalog No. A17108 COX and lipo-oxygenase 抑制剂Timegadine被发现是一种有效的竞争性环加氧酶（COX）和脂加氧酶抑制剂，IC50的范围从5 nM（洗兔血小板）到20μM（大鼠脑）。在马血小板匀浆的细胞溶质级分和洗涤过的兔血小板中，脂氧化酶的浓度为100μM和100μM。 了解更多 -
Aceclofenac
Catalog No. A17433 COX-2 抑制剂Aceclofenac is a cyclooxygenase-2 inhibitor used to treat osteoarthritis, rheumatoid arthritis and ankylosing spondylitis. 了解更多 -
Bromfenac sodium hydrate
Catalog No. A18194 COX-2 抑制剂Bromfenac Sodium Sesquihydrate is a nonsteroidal anti-inflammatory drug (NSAID), which inhibits cyclooxygenase II (COX-2). 了解更多 -
Metamizole sodium hydrate
Catalog No. A18270 COX 抑制剂Dipyrone, also known as Anador and NSC-73205, is a nonsteroidal anti-inflammatory drug used to treat pain (postoperative, colic, cancer, and migraine). 了解更多 -
Ibuprofen (Advil)
Catalog No. A10461 COX-1 抑制剂Ibuprofen (Advil)是一种非甾体抗炎药(NSAID)，靶向COX-1，IC50为13 μM。 了解更多 -
Ibuprofen Lysine (NeoProfen)
Catalog No. A10462 -
Asaraldehyde (Asaronaldehyde)
Catalog No. A10090 -
Celecoxib
Catalog No. A10193 -
Pravadoline (WIN 48098)
Catalog No. A10749 COX 抑制剂Pravadoline (WIN 48098)是抗炎和前列腺素合成抑制剂，通过抑制环氧合酶（COX）发挥作用。 了解更多 -
Sulindac (Clinoril)
Catalog No. A10878 -
Flunixin meglumine
Catalog No. A11686 COX 抑制剂Flunixin Meglumin是一种有效的环氧化酶（COX）抑制剂，用作止痛剂，具有抗炎和解热作用。 了解更多 -
Acemetacin (Emflex)
Catalog No. A11692 -
Tolfenamic acid
Catalog No. A11693 COX-2 抑制剂Tolfenamic Acid是一种COX-2抑制剂，IC50为0.2μM。它是非甾体抗炎药（NSAID）的一类。它用于治疗偏头痛的症状。 了解更多 -
Nimesulide
Catalog No. A11694 -
Lornoxicam (Xefo)
Catalog No. A11695 COX 抑制剂Lornoxicam (Xefo)是一种非甾体类COX-1/COX-2抑制剂。它是oxicam类的非甾体类抗炎药（NSAID），具有镇痛（缓解疼痛），抗炎和退烧（退烧）特性。 了解更多 -
Licofelone
Catalog No. A11697 COX/LOX 抑制剂Licofelone是一种COX/LOX双重抑制剂，被认为是治疗骨关节炎的药物。它可能会降低与其他仅抑制COX（环氧合酶）的非甾体类抗炎药有关的胃肠道毒性。利福非酮是第一种同时抑制两者的药物。 了解更多 -
Diclofenac sodium
Catalog No. A10304 COX 抑制剂Diclofenac Sodium是一种非选择性的COX抑制剂，完整细胞中的COX-1和-2的IC50分别为0.5μg/ml和0.5μg/ml，作用于绵羊COX-1和COX-2， IC50分别为60和220 nM，用作非甾体类抗炎药（NSAID）来减轻疼痛和减轻疼痛 肿胀发炎。 了解更多 -
Iguratimod (T 614)
Catalog No. A11464 COX-2 抑制剂Iguratimod (T 614)是一种抗风湿剂，能够有效地抑制COX-2的活性，IC50值为20 μM (7.7 μg/mL)，而对 COX-1 无作用；Iguratimod同时为巨噬细胞移动抑制因子 (MIF) 抑制剂，IC50值为6.81 μM。 了解更多 -
Piroxicam (Feldene)
Catalog No. A10736 -
Phenylbutazone (Butazolidin, Butatron)
Catalog No. A10720 COX 抑制剂Phenylbutazone (Butazolidin,Butatron)是一种具有研究意义的化合物，它是一种抗炎和抗增殖剂。 了解更多 -
Indomethacin (Indocid, Indocin)
Catalog No. A10474 COX 抑制剂Indomethacin (Indocid, Indocin)是一种非选择性COX1和COX2抑制剂，IC50分别为0.1 μg/mL和5 μg/mL。吲哚美辛(吲哚满，吲哚满)是一种非甾体抗炎药，通常用于减轻发热、疼痛、僵硬和肿胀。 了解更多 -
Rofecoxib (Vioxx)
Catalog No. A11918 -
Eicosatetraynoic acid
Catalog No. A19008 COX/LOX inhibitorEicosatetraynoic acid (ETYA) is a nonspecific inhibitor of cyclooxygenase and lipoxygenase (ID50=8 μM and 4 μM, respectively). Eicosatetraynoic acid (ETYA) activates PPARα and PPARγ chimeras at 10 ?M?? 了解更多 -
Etodolac (AY-24236)
Catalog No. A10371 COX inhibitorEtodolac (AY-24236) is a non-steroidal anti-inflammatory compound that is a non-selective inhibitor of COX (IC50=53.5 nM). 了解更多 -
Naproxen etemesil
Catalog No. A13052 COX-1 and COX-2 inhibitorNaproxen etemesil is a lipophilic, non-acidic, inactive prodrug of naproxen that is hydrolysed to pharmacologically active Naproxen once absorbed. Naproxen is a COX-1 and COX-2 inhibitor with IC50s of 8.72 and 5.15 μM, respectively in cell assay. 了解更多 -
Diclofenac diethylamine
Catalog No. A16503 COX inhibitorDiclofenac diethylamine is a potent and nonselective anti-inflammatory agent, acts as a COX inhibitor. 了解更多 -
Diclofenac
Catalog No. A17814 COX inhibitorDiclofenac is a potent and nonselective anti-inflammatory agent, acts as a COX inhibitor, with IC50s of 4 nM, 1.3 nM for human COX-1 and COX-2 in CHO cells, and 5.1, 0.84 μM for ovine COX-1 and COX-2, respectively. 了解更多 -
Tepoxalin
Catalog No. A12879 -
Etoricoxib D4
Catalog No. A21877 COX-2 inhibitorEtoricoxib D4 (MK-0663 D4) is a deuterium labeled Etoricoxib. Etoricoxib is a non steroidal anti-inflammatory agent, acting as a selective and orally active COX-2 inhibitor, with IC50s of 1.1 μM and 116 μM for COX-2 and COX-1 in human whole blood. 了解更多 -
Fexofenadine HCl
Catalog No. A11859 COX 抑制剂/histamine H1 receptor 激动剂Fexofenadine Hydrochloride是一种抗组胺药，可抑制Cox-1，Cox-2，并且是组胺H1受体激动剂，IC50为246 nM。 了解更多
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