DNA-PK

Catalog No.Inhibitor Name DNA-PKOther
A10726PI-103
**
p110α,p110δ,p110β
A11098NU7441
***
mTOR,PI3K
A10729PIK-75
****
p110α,p110γ,p110δ
A12752NU7026
*
PI3K
A11207PP121
**
PDGFR,Hck,VEGFR
A13224KU-0060648
***
PI3Kδ,PI3Kβ,PI3Kα
A11778Compound 401
*
mTOR,PI3K
A13328ETP-46464
***
ATM, ATR, PI3Kα, mTOR
A15779CC-115
***
mTOR

Notes:
1.Hover mouse over " * " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " * " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.

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  1. PIK-75 hydrochloride

    Catalog No. A10729
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    PI3K 抑制剂
    PIK-75是一种p110α抑制剂,IC50值为5.8nM。在p110γ和p110β的效果较差,IC50值为0.076 ?M和1.3 ?M。 了解更多

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