EGFR/HER2

Inhibitory Selectivity

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Catalog No.	Inhibitor Name	EGFR/ErbB1	HER2/ErbB2	ErbB4	Other
A10043	AEE788	****	***	*	MEK,LCK,VEGFR2
A10047	AG-490	*	*		JAK2
A10053	Tyrphostin AG 879		*		Trk
A10116	Sapitinib	***	***		HDAC,HDAC1,HDAC6
A10141	Afatinib	****	**
A10210	Chrysophanic Acid
A10211	Canertinib	****	***
A10242	CP-724714		**
A10246	CUDC-101	***	**
A10286	Daphnetin	*			PKC, PKA

Showing 1 to 10 of 50 entries

Notes:
1.Hover mouse over " * " to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of " * " is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.