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￥ 0.00 JNK/c-Jun
| Catalog No. | Inhibitor Name | JNK1 | JNK2 | JNK3 | JNK | Other |
|---|---|---|---|---|---|---|
| A10860 | SP600125 | *** | *** | * | Aurora A,TrkA,FLT3 | |
| A12749 | JNK-IN-8 | **** | *** | **** | Kit (V559D,T670I),Kit (V559D),RIOK2 | |
| A11969 | JNK Inhibitor IX | * | ** | |||
| A11296 | AS 602801 (Bentamapimod) | ** | ** | * | ||
| A13564 | CC-930 ( Tanzisertib) | ** | *** | **** | ||
| A13565 | CEP-1347 | *** | ||||
| A13683 | BI-78D3 | * | ||||
| A11352 | CC-401 | |||||
| A15061 | DB07268 | **** | ||||
| A15136 | JNK-IN-7 | IRAK1, PIK3C3, PIP5K3 and PIP4K2C | ||||
| A16036 | IQ 3 | * | * | ** | NF-κB, AP1 | |
| A16039 | SU 3327 | * | ||||
| A16054 | TCS JNK 6o | **** | **** | ** | ||
| A16062 | IQ-1S | * | * | ** | ||
| A15883 | Vacquinol-1 |
Notes:
1.Hover mouse over "" to view the IC50 value.(A few compounds have proven potency but without published IC50 data.)
2.For more details about the compound, click on the product name of your interest.
3.The higher the number of "" is, the more potent the inhibitor or activator is.
4."" refers to compounds which do inhibitory effects on the related isoform, but without specific value.
21 个项目
每页
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JIP-1 (153-163)
Catalog No. A16041 JNK 抑制剂JIP-1 (153-163)是c-Jun N末端激酶（JNK）的肽抑制剂，基于JNK相互作用蛋白1（JIP-1）的153-163残基。以微摩尔范围的亲和力与JNK结合，并最小程度地抑制p38和ERK。 了解更多 -
CC-401 hydrochloride
Catalog No. A15037 -
CEP-1347
Catalog No. A13565 -
CC-930 (Tanzisertib)
Catalog No. A13564 JNK 抑制剂CC-930在蛋白底物c-Jun的JNK依赖性磷酸化中与ATP动力学竞争，并且对JNK的所有同工型均有效（Ki（JNK1）= 44±3 nM，IC50（JNK1）= 61 nM，Ki（JNK2 ）= 6.2±0.6 nM，IC50（JNK2）= 5 nM，IC50（JNK3）= 5 nM），对MAP激酶ERK1和p38a具有选择性，IC50分别为0.48和3.4μM。 了解更多 -
IQ-1S
Catalog No. A16062 -
SR 3576
Catalog No. A16020 -
TCS JNK 5a
Catalog No. A11969 JNK 抑制剂 IXTCS JNK 5a是JNK2和JNK3的高度选择性抑制剂（对于JNK3，JNK2，JNK1和p38β，pIC50值分别为6.7、6.5，<5.0和<4.8）。 了解更多 -
c-JUN peptide
Catalog No. A16045
21 个项目
每页